It is suggested to purchase clomiphene citrate as an agent for a selective action on estrogen receptors. As for estrogen receptors, which are found in the pituitary gland and ovaries, a drug from the triphenylethylene group has a blocking effect.
As a result, the negative feedback mechanism between estrogen and the hypothalamus is hampered. An even more important process takes place along the way: Clomiphene citrate stimulates an increase in the secretion of gonadoliberin by the hypothalamus. As a result, the pituitary gland produces more prolactin, luteinizing hormone, and follicle-stimulating hormone, and testosterone is produced by the testes (testes). Note that the action of the drug does not directly affect the concentration of estrogen in the blood.
What is the significance of the use of the drug
The considered properties of the drug have proven themselves in demand in cases where anabolic androgenic steroids are used. Indeed, as a result of the steroid course, the body greatly reduces the production of natural testosterone, so clomiphene citrate is very important for men. It helps to bring natural testosterone secretion to the required level, which helps to revive sexual activity, increase libido and return to the usual rhythm of sexual activity. Even after the toughest cycles of anabolic androgenic steroids, which seriously affect some body functions, clomiphene citrate successfully copes with the normalization of sexual activity to increase testosterone within two to three months.
As it is suggested to take Clomid as part of post cycle rehabilitation therapy
The drug has a narrow scope. It is used as the main constituent of post-cycle therapy, it begins to be used only after the elimination of the main anabolic androgenic steroids from the body is finished. This is an important prerequisite for using clomiphene and a guarantee of the effectiveness of the effect. Clomiphene citrate, the price of which is significantly higher than that of tamoxifen, which is used for a similar purpose, can be used after any steroid course. This is the advantage over tamoxifen, because post cycle therapy in the case of the use of anabolic androgenic steroids with progestin activity (nandrolones and trenbolones) can only be done with this estrogen receptor blocker (or the rarely used toremifene citrate).
The instructions for use of clomiphene citrate allows such use, since there is no dangerous connection with progesterone receptors in terms of side effects.
Side effects when using the drug
The use of the drug can lead to negative side effects:
- suppression of insulin-like growth factor secretion (IGF-1);
- an increase in the level of globulin that binds sex hormones;
- direct suppression of testicular function;
- a multiple increase in the concentration of estrogen;
- the appearance of a visual impairment (when consumed for a long time.
How Clomiphene Citrate is Used in Bodybuilding
In anticipation of the onset of therapy after the cycle, it is worthwhile to conduct an analysis to determine the actual level of testosterone, and then proceed to restore the optimal functioning of the hypothalamic gland. testicular arch. The duration of recovery therapy is determined by how much the pituitary gland activity has been inhibited. It is usually between two and five weeks.
It does not matter where clomiphene citrate is for sale, in a pharmacy or an online store that provides sports pharmacology products, but there must be confidence in the quality of the medicine purchased.
For an easy course, you should buy the drug in sufficient quantity to take 50 mg for the first two weeks and 25 mg for the next two weeks.
In moderate severity, the duration of daily intake of 50 mg clomid doubled. If you have to take a difficult course of anabolic androgenic steroids, it is worth buying quality Anfarm Hellas clomid, manufactured by a Greek pharmaceutical company founded in 1967. It is taken daily at 100mg for a month, after which the dosage is halved every two weeks .